Fluoroalkylation of porphyrins: synthesis and reactions of beta-fluoroalkyltetraarylporphyrins

Jin, LM; Zeng, Z; Guo, CC; Chen, QY

HERO ID

4923664

Reference Type

Journal Article

Year

2003

Language

English

PMID

12737571

HERO ID 4923664
In Press No
Year 2003
Title Fluoroalkylation of porphyrins: synthesis and reactions of beta-fluoroalkyltetraarylporphyrins
Authors Jin, LM; Zeng, Z; Guo, CC; Chen, QY
Journal Journal of Organic Chemistry
Volume 68
Issue 10
Page Numbers 3912-3917
Abstract Treatment of 5,10,15,20-tetraarylporphyrins (1) with perfluoroalkyl iodides (2) in the presence of Na(2)S(2)O(4)/NaHCO(3) in DMSO-CH(2)Cl(2) at 30-40 degrees C for several hours gives the corresponding 2-perfluoroalkylporphyrins (3). Nucleophilic attack on 3 with dimethyl malonate, diethyl malonate, malonitrile, or cyano acetate (Nu) anion results in the formation of (E)-3-Nu-2-perfuoroalkyl(methylenyl)chlorins. Electrophilic substitution on 3 with NBS or NO(2) affords regioselectively the corresponding 12(or 13)-bromo- and 12,13-dibromo- or nitroporphyrins.
Doi 10.1021/jo0207269
Pmid 12737571
Wosid WOS:000182825000022
Is Certified Translation No
Dupe Override No
Is Public Yes
Language Text English