Palladium-catalyzed enantioselective allylation in the presence of phosphoramidites derived from (S-a)-3-SiMe3-BINOL, (R,S)-semi-TADDOL, and (R,R)-TADDOL

Gavrilov, KN; Zheglov, SV; Novikov, IM; Chuchelkin, IV; Gavrilov, VK; Lugovsky, VV; Zamilatskov, IA

HERO ID

4935985

Reference Type

Journal Article

Year

2015

HERO ID 4935985
In Press No
Year 2015
Title Palladium-catalyzed enantioselective allylation in the presence of phosphoramidites derived from (S-a)-3-SiMe3-BINOL, (R,S)-semi-TADDOL, and (R,R)-TADDOL
Authors Gavrilov, KN; Zheglov, SV; Novikov, IM; Chuchelkin, IV; Gavrilov, VK; Lugovsky, VV; Zamilatskov, IA
Journal Russian Chemical Bulletin
Volume 64
Issue 7
Page Numbers 1595-1601
Abstract Novel P*- and P-monodentate phosphoramidites of a 1,3,2-dioxaphosphepine series were derived from (S-a)-3-trimethylsilyl-BINOL, (R,S)-semi-TADDOL, and (R,R)-TADDOL. Catalytic performance of the synthesized compounds were examined in the Pd-catalyzed asymmetric allylic substitution of (E)-1,3-diphenylallyl acetate: the reaction with dimethyl malonate gave up to 92% ee. The effects of additives of 5,10,15,20-tetraphenylporphyrin and its metal complexes on conversion and enantioselectivity were studied.
Doi 10.1007/s11172-015-1047-7
Wosid WOS:000375794600013
Is Certified Translation No
Dupe Override No
Is Public Yes
Keyword chiral phosphoramidites; palladium catalysts; asymmetric allylation; 5,10,15,20-tetraphenylporphyrin