Fused polycyclic hydrocarbons through superacid-induced cyclialkylation of aromatics

Ledneczki, I; Forgo, P; Molnar, A

HERO ID

857495

Reference Type

Journal Article

Year

2007

Language

English

HERO ID 857495
In Press No
Year 2007
Title Fused polycyclic hydrocarbons through superacid-induced cyclialkylation of aromatics
Authors Ledneczki, I; Forgo, P; Molnar, A
Journal Catalysis Letters
Volume 119
Issue 3-4
Page Numbers 296-303
Abstract Benzene and substituted derivatives (toluene, ortho-xylene, 1,2,3-trimethylbenzene, 1,2,4-trimethylbenzene, anisole), when applied in large excess, react with 1,4 diols (pentan-1,4-diol, hexan-2,5-diol, and 2,5-dimethylhexan-2,5-diol) or an oxolane (2,2,5,5-tetramethyltetrahydrofuran) in the presence of the Bronsted superacid trifluoromethanesulfonic acid (triflic acid, TFSA) to afford substituted tetralins in excellent yields with high selectivity. Reacting benzene with a small excess of alkylating agents yields octahydroanthracenes. The transformation of naphthalene with oxolane leads to a partially saturated octamethyloctahydrotetracene under similar conditions. Product formation is interpreted by intermolecular Friedel-Crafts alkylation followed by cyclialkylative ring closure.
Doi 10.1007/s10562-007-9234-2
Wosid WOS:000250996200016
Url <Go to ISI>://WOS:000250996200016
Is Certified Translation No
Dupe Override No
Is Public Yes
Language Text English
Keyword alkylation; cyclialkylation; arenes; carbocations; superacid; chemistry, physical
Is Qa No