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HERO ID
7418929
Reference Type
Journal Article
Title
Interaction of disulfiram with antiretroviral medications: efavirenz increases while atazanavir decreases disulfiram effect on enzymes of alcohol metabolism
Author(s)
Mccance-Katz, EF; Gruber, VA; Beatty, G; Lum, P; Ma, Q; Difrancesco, R; Hochreiter, J; Wallace, PK; Faiman, MD; Morse, GD; ,
Year
2013
Is Peer Reviewed?
Yes
Journal
American Journal on Addictions
ISSN:
1055-0496
Volume
23
Issue
2
Page Numbers
137-144
Language
English
PMID
24118434
DOI
10.1111/j.1521-0391.2013.12081.x
URL
http://doi.wiley.com/10.1111/j.1521-0391.2013.12081.x
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Abstract
Alcohol abuse complicates treatment of HIV disease and is linked to poor outcomes. Alcohol pharmacotherapies, including disulfiram (DIS), are infrequently utilized in co-occurring HIV and alcohol use disorders possibly related to concerns about drug interactions between antiretroviral (ARV) medications and DIS.
Keywords
alcohol; aldehyde dehydrogenase; anti human immunodeficiency virus agent; atazanavir; benzoxazine derivative; diethyldithiocarbamic acid; disulfiram; drugs used in the treatment of addiction; efavirenz; oligopeptide; pyridine derivative; ritonavir; S-methyl diethylthiocarbamate; S-methyl N,N-diethylthiolcarbamate sulfoxide; thiocarbamic acid derivative; adult; agonists; alcoholism; analogs and derivatives; antagonists and inhibitors; biotransformation; clinical trial; combination drug therapy; drug effects; drug interaction; female; half life time; human; male; metabolism; middle aged; normal human; Adult; Alcohol Deterrents; Alcoholism; Aldehyde Dehydrogenase; Anti-HIV Agents; Atazanavir Sulfate; Benzoxazines; Biotransformation; Disulfiram; Ditiocarb; Drug Interactions; Drug Therapy, Combination; Ethanol; Female; Half-Life; Healthy Volunteers; Humans; Male; Middle Aged; Oligopeptides; Pyridines; Ritonavir; Thiocarbamates
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