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7560621 
Journal Article 
Anilines Made Easily: From Aldehydes to Tri-, Tetra-, and Pentasubstituted Anilines in Two Steps 
Neumann, H; Jacobi von Wangelin, A; Klaus, S; Strübing, D; Gördes, D; Beller, M; , 
2003 
Yes 
Angewandte Chemie (International Edition)
ISSN: 1433-7851
EISSN: 1521-3773 
WILEY-V C H VERLAG GMBH 
WEINHEIM 
42 
37 
4503-4507 
English 
Easy as one, two, three. Highly substituted anilines are accessible with unprecedented efficiency from the three-component-coupling reaction of O-benzyl carbamate, aldehydes, and dienophiles followed by a new domino aromatization/deprotection reaction involving transfer hydrogenation (see scheme). EWG: electron-withdrawing group. 
Anilines; Multicomponent reactions; Palladium; Transfer hydrogenation; Aldehydes; Amines; Aromatization; Hydrogenation; Reaction kinetics; Synthesis (chemical); Transfer hydrogenation; Aromatic compounds; aldehyde; aniline derivative; carbamic acid derivative; o benzyl carbamate; unclassified drug; aromatization; article; chemical reaction; chemical structure; deprotection reaction; electron; hydrogenation; reaction analysis; structure analysis; synthesis; three component coupling reaction